AN EFFICIENT SYNTHESIS OF 3'-FLUORO-3'-DEOXYTHYMIDINE (FLT)

被引：26

作者：

HAGER, MW ^{[1
]}

LIOTTA, DC ^{[1
]}

机构：

[1] EMORY UNIV,DEPT CHEM,ATLANTA,GA 30322

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 47期

基金：

美国国家卫生研究院;

关键词：

D O I：

10.1016/S0040-4039(00)60841-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A synthetic route which permits the regioselective introduction of fluoride into an FLT precursor under mild conditions and the subsequent conversion of that intermediate into FLT is reported.

引用

页码：7083 / 7086

页数：4

共 16 条

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