Ruthenium-Catalyzed Direct C-H Bond Arylations of Heteroarenes

被引：256

作者：

Ackermann, Lutz ^{[1
]}

Lygin, Alexander V. ^{[1
]}

机构：

[1] Univ Gottingen, Inst Organ & Biomol Chem, D-37077 Gottingen, Germany

来源：

ORGANIC LETTERS | 2011年 / 13卷 / 13期

关键词：

RH(I)-CATALYZED DIRECT ARYLATION; AZOLE N-OXIDES; CARBON-HYDROGEN; PHOSPHINE OXIDES; PALLADIUM; FUNCTIONALIZATION; HETEROCYCLES; INDOLES; PRELIGANDS; ARENES;

D O I：

10.1021/ol2010648

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Ruthenium-catalyzed C-H bond arylations of indoles, thiophenes, and pyrroles were accomplished in a highly chemo- and site-selective manner through the use of removable directing groups.

引用

页码：3332 / 3335

页数：4

共 77 条

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