Solid-phase organic reactions .2. A review of the literature Nov 95 Nov 96.

被引:439
作者
Hermkens, PHH [1 ]
Ottenheijm, HCJ [1 ]
Rees, DC [1 ]
机构
[1] ORGANON LABS,SCI DEV GRP,NEWHOUSE ML1 5SH,SCOTLAND
关键词
D O I
10.1016/S0040-4020(97)00279-2
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
This Report reviews literature published Nov 1995-Nov 1996 and summarises organic reactions performed on solid-supports. The reactions are presented in a graphical abstract format and examples of amide formation, aromatic nucleophilic substitution, cleavage, condensation, cycloaddition, deprotection, Grignard, heterocycle formation, immobilisation to resin, Michael addition, miscellaneous, multiple component condensation, olefin formation, oxidation, reduction and substitution (nucleophilic/electrophilic) are given. The review is designed as an update to Tetrahedron Report no. 394. (C) 1997 Elsevier Science Ltd.
引用
收藏
页码:5643 / 5678
页数:36
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